MOR agonist-1
MOR agonist-1 is a MOR (μ-opioid receptor) agonist. MOR agonist-1 has good analgesic effect. MOR agonist-1 can be used for the research of pain and pain-related disorders.
For research use only. We do not sell to patients.
- CAS No.: 2305781-14-8
- Formula: C22H26ClFN2O2
- Molecular Weight:404.91
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Opioid Receptor Isoforms
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Biological Activity
MOR agonist-1 has cAMP agonist activity for human μ-subtype opioid receptors (hMOR) with an EC50 value of o.5 nM[1].
MOR agonist-1 has inhibitory activity for CYP2C19, CYP2D6 and CYP3A4 with IC50 values of 33.7 μM, 12.7 μM and 40.6 μM, respectively[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2305781-14-8
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Molecular Weight 404.91
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Formula C22H26ClFN2O2
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SMILES
ClC1=CC=CC(CNCC[C@]2(C3=CC=C(C=N3)F)C[C@@]4(CCOC4)OCC2)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)