MRS-1706 (Standard)
MRS-1706 (Standard) is the analytical standard of MRS-1706. This product is intended for research and analytical applications. MRS-1706 is a potent and selective adenosine A2B receptor inverse agonist. MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1 and A3 receptors respectively. MRS-1706 blocks adenosine-mediated cAMP induction.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- Purity : 95%
- CAS No.: 264622-53-9
- 화학식: C27H29N5O5
- 분자량:503.55
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보관:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Product Information
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Chemical Information
- 순도&문서
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Help & FAQs
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HY-103186
MRS-1706Adenosine A2B Inverse Agonist -
HY-103173
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SCH 58261A2A Receptor Antagonist -
HY-14121
MRS 1754A2B Antagonist -
HY-13201
CGS 21680 -
HY-13201A
CGS 21680 HydrochlorideAdenosine A2A Receptor Agonist -
HY-19532
ZM241385A2A Receptor Antagonist -
HY-123085
AlloxazineA2b Antagonist -
HY-10888
IstradefyllineAdenosine A2A Receptor Antagonist -
HY-103171
BAY 60-6583A2B Receptor Agonist -
HY-100937
DPCPXA1 Receptor Antagonist -
HY-103166
PSB-603A2B Receptor Antagonist
Product Information
Information
신청
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
Chemical Information
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CAS No. 264622-53-9
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분자량 503.55
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화학식 C27H29N5O5
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SMILES
O=C(NC1=CC=C(C(C)=O)C=C1)COC2=CC=C(C3=NC(N(CCC)C(N(CCC)C4=O)=O)=C4N3)C=C2
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
[1]. Li Q, et, al. ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor. J Pharmacol Exp Ther. 2007 Feb;320(2):637-45. [Content Brief]
[2]. Mi T, et, al. Excess adenosine in murine penile erectile tissues contributes to priapism via A2B adenosine receptor signaling. J Clin Invest. 2008 Apr;118(4):1491-501. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MRS-1706 (Standard) Related Classifications
HY-103186R Related Classifications
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