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Referencia número: HY-P1292A

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PKG inhibitor peptide TFA

Name: PKG inhibitor peptide TFA
Brand: MedChemExpress
SKU: HY-P1292A
Availability: PreOrder

2 Cited Publications

Revisión del cliente

Based on 2 publication(s) in Google Scholar

PKG inhibitor peptide TFA is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a K_i of 86 μM.

Para uso exclusivo en investigación. No vendemos a pacientes.

Fòrmula: C₄₀H₇₅F₃N₁₈O₁₂
Peso molecular:1057.13

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

PKG inhibitor peptide TFA Chemical Structure

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica
- Descripciòn
- IC₅₀ & Target
- In Vitro
Chemical Information
Publications (2)
Pureza y Documentación
Referencias
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Bioz

Actividad biológica

Descripciòn

PKG inhibitor peptide TFA is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a K_i of 86 μM^[1].

IC₅₀ & Target

Ki: 86 μM (PKG)^[1]

In Vitro

Summary of experiments showing that intracellular dialysis of postsynaptic cells with PKG inhibitor PKG inhibitor peptide TFA (1 mM) failed to alter the induction of long-term depression (CCh-LTD)^[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

Peso molecular 1057.13
Fòrmula C₄₀H₇₅F₃N₁₈O₁₂
Sequence

Arg-Lys-Arg-Ala-Arg-Lys-Glu
Sequence Shortening

RKRARKE
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Publications (2)

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Nature

Rescuing dendritic cell interstitial motility sustains antitumour immunity. [Abstract]

2025 Sep;645(8079):244-253. PMID: 40562926
Oncogene

LAMP5 modulates IRF4 stability and nuclear transport: a critical mechanism in myeloma progression and therapy. [Abstract]

2025 Jul 28. PMID: 40721659

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (258 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Bhatnagar D, et al. Synthetic peptide analogues differentially alter the binding affinities of cyclic nucleotide dependent protein kinases for nucleotide substrates. Biochemistry. 1988 Mar 22;27(6):1988-94. [Content Brief]

[2]. Chiung-Chun Huang, et al. Activation of muscarinic acetylcholine receptors induces a nitric oxide-dependent long-term depression in rat medial prefrontal cortex. Cereb Cortex. 2010 Apr;20(4):982-96. [Content Brief]

Calculators

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

PKG inhibitor peptide TFA

2 Cited Publications

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Actividad biológica
- Descripciòn
- IC₅₀ & Target
- In Vitro
Chemical Information
Publications (2)
Pureza y Documentación
Referencias

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PKG inhibitor peptide TFA

Publications Citing Use of MedChemExpress (MCE) PKG inhibitor peptide TFA