rel-Asenapine hydrochloride
rel-Asenapine (rel-Org 5222) hydrochloride is a relative configuration of Asenapine hydrochloride (HY-16567). Asenapine (Org 5222) hydrochloride, an atypical antipsychotic, is an antagonist of serotonin receptors (pKi: 8.4-10.5), adrenoceptors (pKi: 8.9-9.5), dopamine receptors (pKi: 8.9-9.4) and histamine receptors (pKi: 8.2-9.0). Asenapine hydrochloride can be used in the research of schizophrenia and bipolar disorder.
For research use only. We do not sell to patients.
- CAS No.: 1261398-77-9
- Formula: C17H17Cl2NO
- Molecular Weight:322.23
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All 5-HT Receptor Isoforms
MoreAll Adrenergic Receptor Isoforms
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Biological Activity
Chemical Information
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CAS No. 1261398-77-9
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Molecular Weight 322.23
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Formula C17H17Cl2NO
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SMILES
CN1C[C@@]2([H])[C@@](C1)([H])C3=CC=CC=C3OC4=CC=C(Cl)C=C42.Cl
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Synonyms
rel-Org 5222 hydrochloride
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Shahid M, et al. Asenapine: a novel psychopharmacologic agent with a unique human receptor signature. J Psychopharmacol. 2009 Jan;23(1):65-73. [Content Brief]
[2]. Olivia Frånberg, et al. Asenapine, a novel psychopharmacologic agent: preclinical evidence for clinical effects in schizophrenia. Psychopharmacology (Berl). 2008 Feb;196(3):417-29. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)