RESA peptide
Based on 1 Customer Validation
RESA peptide is a substrate peptide of β-adrenergic receptor kinase (βARK). RESA peptide serves as a substrate for βARK-mediated phosphorylation, and its N-terminal acidic residues enhance phosphorylation efficiency and substrate binding capacity.
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- Purity: 99.97%
- CAS No.: 133699-13-5
- 화학식: C55H93N21O24
- 분자량:1432.45
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보관:
Sealed storage, away from moisture.
Powder -80°C, 2 years , -20°C, 1 year* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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용액&용해도
- 순도&문서
- References
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Help & FAQs
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Biological Activity
The RESA peptide (RRREEEEESAAA) (0.05-7 mM; 60 min) acts as a substrate for purified βARK1 with a Vmax/Km ratio of 39, which is 240-fold higher than the basic peptide RRRASAAASAA and ~4000-fold lower than activated rhodopsin[1].
The RESA peptide (RRREEEEESAAA) (0.05-3 mM; 60 min) had its βARK1-mediated phosphorylation slightly inhibited by light-activated rhodopsin (Rho'), reducing the Vmax/Km ratio to 0.6-fold of the value measured in the absence of Rho'[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 133699-13-5
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Appearance Solid
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분자량 1432.45
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화학식 C55H93N21O24
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Color White to off-white
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Sequence
Arg-Arg-Arg-Glu-Glu-Glu-Glu-Glu-Ser-Ala-Ala-Ala
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Sequence Shortening
RRREEEEESAAA
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Sealed storage, away from moisture
Powder -80°C 2 years -20°C 1 year * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
용액&용해도
DMSO : 100 mg/mL (69.81 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
순도&문서
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Data Sheet (271 KB)
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SDS (254 KB)
- English - EN (254 KB)
- Français - FR (254 KB)
- Deutsch - DE (254 KB)
- Norwegian - NO (254 KB)
- Español - ES (254 KB)
- Swedish - SV (254 KB)
- Italian - IT (254 KB)
- Korean - KR (254 KB)
- Portuguese - PT (254 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 0.6981 mL | 3.4905 mL | 6.9810 mL | 17.4526 mL |
| 5 mM | 0.1396 mL | 0.6981 mL | 1.3962 mL | 3.4905 mL | |
| 10 mM | 0.0698 mL | 0.3491 mL | 0.6981 mL | 1.7453 mL | |
| 15 mM | 0.0465 mL | 0.2327 mL | 0.4654 mL | 1.1635 mL | |
| 20 mM | 0.0349 mL | 0.1745 mL | 0.3491 mL | 0.8726 mL | |
| 25 mM | 0.0279 mL | 0.1396 mL | 0.2792 mL | 0.6981 mL | |
| 30 mM | 0.0233 mL | 0.1164 mL | 0.2327 mL | 0.5818 mL | |
| 40 mM | 0.0175 mL | 0.0873 mL | 0.1745 mL | 0.4363 mL | |
| 50 mM | 0.0140 mL | 0.0698 mL | 0.1396 mL | 0.3491 mL | |
| 60 mM | 0.0116 mL | 0.0582 mL | 0.1164 mL | 0.2909 mL |
RESA peptide Related Classifications
HY-P11765 Related Classifications
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