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Cat. No.: HY-164037

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Riselcaftor

Riselcaftor (Example 33) is a CFTR modulator, with an EC₅₀ of 20.1 nM in human bronchial epithelial cells. Riselcaftor can be used for research of cystic fibrosis.

For research use only. We do not sell to patients.

CAS No.: 2799652-36-9
Formula: C₂₉H₂₈N₂O₅S
Molecular Weight:516.61

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

Riselcaftor Chemical Structure

CAS No.: 2799652-36-9

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Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

Riselcaftor (Example 33) is a CFTR modulator, with an EC₅₀ of 20.1 nM in human bronchial epithelial cells. Riselcaftor can be used for research of cystic fibrosis^[1].

Chemical Information

CAS No. 2799652-36-9
Molecular Weight 516.61
Formula C₂₉H₂₈N₂O₅S
SMILES

O=S(NC([C@]1(C2=C(C=CC(C)=C2)OC)C[C@H](C3=CC=CC=C3)CO1)=O)(C4=CC=CC5=C4C=CC(C)=N5)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. David J. Hardee, et al. Modulators of the Cystic Fibrosis Transmembrane Conductance Regulator Protein and Methods of Use. Patent. US20220211692 A1

Calculators

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

100 mg

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