RSK2-IN-2
RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 (RSK2) kinase. RSK2-IN-2 is also described to inhibit MSK1, MSK2 and RSK3.
For research use only. We do not sell to patients.
- CAS No.: 1637749-78-0
- Formula: C16H11N5O
- Molecular Weight:289.29
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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RSK2 |
RSK3 |
MSK1 |
MSK2 |
RSK2-IN-2 (Compound 25) shows strong activity with ERK2-MSK1 cascade pIC50 of 9.6[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 1637749-78-0
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Molecular Weight 289.29
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Formula C16H11N5O
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SMILES
O=C(N)/C(C#N)=C/C1=CC=CC(C2=C3C(NC=C3)=NC=N2)=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
RSK2-IN-2 Related Classifications
HY-150643 Related Classifications
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