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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
30 Results for "
congeners
" in MedChemExpress (MCE) Product Catalog:
Products (30)
30 Results for "congeners" in MCE Product Catalog:
1
Target:
Domaines de recherche:
Adenosine amine congener (ADAC) is a selective A1 adenosine receptor agonist, can ameliorate noise- and Cisplatin-induced cochlear injury. Adenosine amine congener also has neuroprotective effects .
1
1 Cited Publications
Synonyms: XAC hydrochloride
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Domaines de recherche:
Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist. Xanthine amine congener hydrochloride induces convulsions in mice .
Cat. No.: HY-N0685
CAS No.: 55954-61-5
Category:
Infection Quinones Anthraquinones Guttiferae Extract Hyperlcurn perforatum L. Phenols Polyphenols Plants Disease Research Fields
Target:
Cat. No.: HY-W013788
CAS No.: 23470-00-0
Synonyms: 2-Palm-Gl
Target:
Cat. No.: HY-118816
CAS No.: 714966-38-8
Synonyms: 11-epi PGF2α-EA; 11β-PGF2α-EA; 11β-Prostamide F2α
Target:
Domaines de recherche:
11β-Prostaglandin F2α ethanolamide (11β-PGF2α-EA) is the theoretical hepatic metabolite of PGD2-EA, produced during COX-2 metabolism of the endogenous cannabinoid AEA which is found in brain, liver, and other mammalian tissues.1 AEA can be used directly by COX-2 and specific PG synthase to produce ethanolamide congeners of the classical PGs. PGD2-EA is formed in activated RAW 264.7 cells treated with AEA.
Cat. No.: HY-101139
CAS No.: 96865-92-8
Synonyms: XAC
Target:
Domaines de recherche:
Xanthine amine congener is a non-selective adenosine receptor antagonist . Xanthine amine congener induces convulsions in mice .
Cat. No.: HY-144286
CAS No.: 2761009-43-0
CXCR4 antagonist 3 (compound 12a) is a potent antagonist of CXCR4 with an IC50 of 11 nM. CXCR4 antagonist 3 is a congener of TIQ15. CXCR4 antagonist 3 demonstrates the best overall properties including CXCR4 antagonism, CYP 2D6 inhibition, metabolic stability, and permeability. CXCR4 antagonist 3 has the potential for the research of human immunodeficiency virus .
Cat. No.: HY-101139AR
CAS No.: 1783977-95-6
Synonyms: XAC hydrochloride (Standard)
Domaines de recherche:
Xanthine amine congener (hydrochloride) (Standard) is the analytical standard of Xanthine amine congener (hydrochloride). This product is intended for research and analytical applications. Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist. Xanthine amine congener hydrochloride induces convulsions in mice .
Cat. No.: HY-110303
CAS No.: 1962928-23-9
Synonyms: XAC dihydrochloride
Target:
Domaines de recherche:
Xanthine amine congener dihydrochloride (XAC dihydrochloride) is a potent Adenosine A1 receptor and A2 receptor antagonist with IC50 values of 1.8 and 114 nM, respectively. Xanthine amine congener acts as a convulsant agent in mice model .
Cat. No.: HY-105890
CAS No.: 74790-08-2
Synonyms: TNO 6
Domaines de recherche:
Spiroplatin is a Cisplatin (HY-17394) congener and has antitumor activity .
Cat. No.: HY-146970
Target:
Domaines de recherche:
Lankacyclinone C is a lankacidin C congener lacking the δ-lactone moiety, with antitumor activity .
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Domaines de recherche:
Fenethazine (Phenethazine) is a compound with antihistamine activity. It is an effective antihistamine. Its congeners also have anticholinergic effects and can be used to inhibit Parkinson's disease.
Cat. No.: HY-N0449R
CAS No.: 28789-35-7
Category:
Alkaloids Capsicum annuum L. Monophenols Other Alkaloids Phenols Plants Solanaceae Extract
Target:
Cat. No.: HY-117765
CAS No.: 129173-57-5
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Domaines de recherche:
RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction .
Cat. No.: HY-148649
CAS No.: 41089-03-6
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Domaines de recherche:
Demethyl bleomycin A2 is a Bleomycin (HY-108345) congener. The DNA cleavage of demethyl bleomycin A2 is insensitive to the presence of 5-Methylcytidine (HY-113135) .
Cat. No.: HY-N0685R
CAS No.: 55954-61-5
Category:
Quinones Anthraquinones Guttiferae Extract Hyperlcurn perforatum L. Phenols Polyphenols Plants
Target:
Cat. No.: HY-N12760
CAS No.: 1800562-59-7
Category:
Target:
Target:
Domaines de recherche:
N-Methylindan-2-amine hydrochloride (compound 3b) is an N-alkylated congener of phenylethylamine that increases hot plate reaction time in mice without inducing dopaminergic effects. N-Methylindan-2-amine hydrochloride can be used to study central noradrenergic mechanisms .
Cat. No.: HY-146102
CAS No.: 2479356-53-9
M1 ligand 1 (compound 3b-b) is a muscarinic acetylcholine receptor M1 ligand. M1 ligand 1 is a N-desmethyl congener of arecoline derivative. M1 ligand 1 can be used as PET (positron emission tomography) radiotracer .
Cat. No.: HY-129454
CAS No.: 485815-59-6
Synonyms: Antibiotic TPU-0037-A
Target:
Domaines de recherche:
TPU-0037A is an antibiotic and a congener of lydicamycin. It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs=1.56-12.5 μg/mL), but not Gram-negative E. coli, P. mirabilis, P. vulgaris, or P. aeruginosa strains (MICs=>50 μg/mL).
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
