TG2-IN-3h
TG2-IN-3h (Compound 3h) is a transglutaminase (TG2) inhibitor (hTG2: IC50 = 6nM). TG2-IN-3h inhibits endothelial cell migration and angiogenesis. TG2-IN-3h alleviates renal fibrosis in a mouse model of hypertensive nephropathy. TG2-IN-3h can be used in research on metabolic diseases such as hypertensive nephropathy and cardiovascular and cerebrovascular diseases such as pathological angiogenesis.
For research use only. We do not sell to patients.
- CAS No.: 1592640-75-9
- Formula: C21H26N4O4S
- Molecular Weight:430.52
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 1592640-75-9
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Molecular Weight 430.52
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Formula C21H26N4O4S
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SMILES
O=C(C=C)NCC(=O)N1CCN(CC1)S(=O)(=O)C2=CC=CC=3C2=CC=CC3N(C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)