TP-680
TP-680 is a cholecystokinin receptor antagonist. TP-680 binds 1510 times more strongly to rat pancreatic CCKA receptors (IC50=1.2 nM) than to rat brain CCKB receptors (IC50=1812.5 nM). TP-680 can be used in the study of gastrointestinal diseases.
For research use only. We do not sell to patients.
- CAS No.: 176915-07-4
- Formula: C35H33N5O4S
- Molecular Weight:619.73
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
CCKAR 1.2 nM (IC50) |
CCKBR 1812.5 nM (IC50) |
Chemical Information
-
CAS No. 176915-07-4
-
Molecular Weight 619.73
-
Formula C35H33N5O4S
-
SMILES
O=C(O)C1=CC=CN=C1SC[C@@H](C(N2CCN(CC2)C(C3=CC=CC=C3)C4=CC=CC=C4)=O)NC(C5=CC6=C(C=CC=C6)N5)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Powered by Bioz