1. Membrane Transporter/Ion Channel
  2. Potassium Channel
  3. VU0134992

VU0134992 

Cat. No.: HY-122560
Handling Instructions

VU0134992 is a selective inward rectifier potassium (Kir) channel Kir4.1 blocker with an IC50 of 0.97 µM.

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VU0134992 Chemical Structure

VU0134992 Chemical Structure

CAS No. : 755002-90-5

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Description

VU0134992 is a selective inward rectifier potassium (Kir) channel Kir4.1 blocker with an IC50 of 0.97 µM[1].

IC50 & Target

IC50: 0.97 µM (Kir4.1)[1]

In Vitro

VU0134992 is greater than 30-fold selective for Kir4.1 over Kir1.1, Kir2.1, and Kir2.2, is weakly active toward Kir2.3, Kir6.2/SUR1, and Kir7.1, and is equally active toward Kir3.1/3.2, Kir3.1/3.4, and Kir4.2[1].

Molecular Weight

411.38

Formula

C₂₀H₃₁BrN₂O₂

CAS No.

755002-90-5

SMILES

O=C(NC1CC(C)(C)NC(C)(C)C1)COC2=CC=C(C(C)C)C=C2Br

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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VU0134992
Cat. No.:
HY-122560
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