1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. nAChR
  3. 3-Bromocytisine

3-Bromocytisine (Synonyms: 3-Br-cytisine)

Cat. No.: HY-107684
Handling Instructions

3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC50s are 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively.

For research use only. We do not sell to patients.

3-Bromocytisine Chemical Structure

3-Bromocytisine Chemical Structure

CAS No. : 207390-14-5

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Description

3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC50s are 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively[1][2].

IC50 & Target

IC50: 0.28 nM (hα4β4), 0.30 nM (hα4β2), 31.6 nM (hα7)[1]

Molecular Weight

269.14

Formula

C₁₁H₁₃BrN₂O

CAS No.

207390-14-5

SMILES

O=C1N2C([[email protected]]3([H])C[[email protected]](CNC3)([H])C2)=CC=C1Br

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

3-Bromocytisine3-Br-cytisinenAChRNicotinic acetylcholine receptorsInhibitorinhibitorinhibit

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3-Bromocytisine
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