1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Neuropeptide Y Receptor
  4. NPY Y1 receptor Isoform
  5. NPY Y1 receptor Antagonist

NPY Y1 receptor Antagonist

NPY Y1 receptor Antagonists (5):

Cat. No. Product Name Effect Purity
  • HY-107726
    BIBP3226 TFA
    Antagonist 98.55%
    BIBP3226 TFA is a potent and selective neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor antagonist, with Kis of 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF, respectively. BIBP3226 TFA displays anxiogenic-like effect.
  • HY-107382
    RF9
    Antagonist 98.04%
    RF9 is a potent and selective Neuropeptide FF receptor antagonist, with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
  • HY-107382A
    RF9 hydrochloride
    Antagonist 99.91%
    RF9 hydrochloride is a potent and selective Neuropeptide FF receptor antagonist, with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
  • HY-107733
    NTNCB hydrochloride
    Antagonist 98.07%
    NTNCB (Compound 11) hydrochloride is a potent and selective neuropeptide Y Y5 (NPY Y5) receptor antagonist with a Ki of 8 nM against human Y5.
  • HY-144603
    Neuropeptide Y Y1 receptor antagonist 1
    Antagonist
    Neuropeptide Y Y1 receptor antagonist 1 (compound 39), a fluorescent probe, is a potent antagonist of neuropeptide Y Y1 receptor (Y1R), with a Ki of 0.19 nM.