1. GPCR/G Protein
    Neuronal Signaling
  2. Melatonin Receptor

Tasimelteon (Synonyms: BMS-214778; VEC-162)

Cat. No.: HY-14803 Purity: 99.92%
Handling Instructions

Tasimelteon is a melatonin MT1 and MT2 receptor agonist.

For research use only. We do not sell to patients.

Tasimelteon Chemical Structure

Tasimelteon Chemical Structure

CAS No. : 609799-22-6

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 66 In-stock
Estimated Time of Arrival: December 31
5 mg USD 60 In-stock
Estimated Time of Arrival: December 31
10 mg USD 90 In-stock
Estimated Time of Arrival: December 31
50 mg USD 290 In-stock
Estimated Time of Arrival: December 31
100 mg USD 490 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Technical Information

  • Purity & Documentation

  • References

Description

Tasimelteon is a melatonin MT1 and MT2 receptor agonist. Target: melatonin receptor Tasimelteon is a novel circadian regulator, is the first product for the treatment of Non-24-hour Sleep-Wake Disorder (Non-24) approved by either the FDA or the European Medicines Agency (EMA). Tasimelteon is a potent and specific melatonin (MT1 and MT2) receptor agonist with 2 - 4 times greater affinity for the MT2 receptor.

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : ≥ 33 mg/mL (134.52 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 4.0763 mL 20.3815 mL 40.7631 mL
5 mM 0.8153 mL 4.0763 mL 8.1526 mL
10 mM 0.4076 mL 2.0382 mL 4.0763 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

245.32

Formula

C₁₅H₁₉NO₂

CAS No.

609799-22-6

SMILES

[H][[email protected]]1(C2=C3C(OCC3)=CC=C2)[[email protected]@](CNC(CC)=O)([H])C1

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country or Region *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Tasimelteon
Cat. No.:
HY-14803
Quantity:

Tasimelteon

Cat. No.: HY-14803