1. GPCR/G Protein
    Neuronal Signaling
  2. Melatonin Receptor

Tasimelteon (Synonyms: BMS-214778; VEC-162)

Cat. No.: HY-14803 Purity: 99.92%
Handling Instructions

Tasimelteon is a melatonin MT1 and MT2 receptor agonist.

For research use only. We do not sell to patients.

Tasimelteon Chemical Structure

Tasimelteon Chemical Structure

CAS No. : 609799-22-6

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 66 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
5 mg USD 60 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
10 mg USD 90 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
50 mg USD 290 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
100 mg USD 490 In-stock
Stock in Sweden
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Related Small Molecules:

  • Biological Activity

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  • Purity & Documentation

  • References

Description

Tasimelteon is a melatonin MT1 and MT2 receptor agonist. Target: melatonin receptor Tasimelteon is a novel circadian regulator, is the first product for the treatment of Non-24-hour Sleep-Wake Disorder (Non-24) approved by either the FDA or the European Medicines Agency (EMA). Tasimelteon is a potent and specific melatonin (MT1 and MT2) receptor agonist with 2 - 4 times greater affinity for the MT2 receptor.

Clinical Trial
References
Preparing Stock Solutions
Concentration Volume Mass 1 mg 5 mg 10 mg
1 mM 4.0763 mL 20.3815 mL 40.7631 mL
5 mM 0.8153 mL 4.0763 mL 8.1526 mL
10 mM 0.4076 mL 2.0382 mL 4.0763 mL
Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

245.32

Formula

C₁₅H₁₉NO₂

CAS No.

609799-22-6

SMILES

[H][[email protected]]1(C2=C3C(OCC3)=CC=C2)[[email protected]@](CNC(CC)=O)([H])C1

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

DMSO: ≥ 33 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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Product Name:
Tasimelteon
Cat. No.:
HY-14803
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