LY-395153
LY-395153 is an AMPA receptor enhancer with the activity of binding to AMPA receptors. LY-395153 can bind to natural and recombinant AMPA receptors, and its binding is affected by AMPA receptor agonists and can be competitively or non-competitively inhibited by some compounds. It is a useful probe for marking unique regulatory sites of AMPA receptors.
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- CAS. Nr.: 211313-51-8
- Formel: C19H24N2O3S
- Molecular Weight:360.47
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
Beschreibung
Cellular Effect
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
0.52 μM
Compound: 24
|
Inhibition of GluR4 expressed in HEK293 cells
Inhibition of GluR4 expressed in HEK293 cells
|
[PMID: 20839777] |
Chemical Information
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CAS. Nr. 211313-51-8
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Molecular Weight 360.47
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Formel C19H24N2O3S
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SMILES
O=C(C1=CC=CC=C1)NC2=CC=C(C(CNS(=O)(C(C)C)=O)C)C=C2
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)