BN-81674
BN-81674 is a somatostatin analogue and a selective antagonist of the non-peptide human somatostatin sst3 receptor (Ki=0.92 nM). In addition, BN-81674 reversed the inhibition of cyclic AMP accumulation induced by 1 nM somatostatin through the sst3 receptor with an IC50 value of 0.84 nM. BN-81674 can be used in cancer research.
For research use only. We do not sell to patients.
- CAS No.: 252278-73-2
- Formula: C30H38N4
- Molecular Weight:454.65
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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SSTR3 0.92 nM (Ki) |
Chemical Information
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CAS No. 252278-73-2
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Molecular Weight 454.65
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Formula C30H38N4
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SMILES
CCCCCC1(N[C@H](CC2=C1NC3=C2C=CC=C3)C4=NC=C(N4)C5=CC=CC=C5)CCCCC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)