BX430 (Standard)
BX430 (Standard) is the analytical standard of BX430 (HY-110237). This product is intended for research and analytical applications. BX430 is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonist with an IC50 of 0.54 μM. BX430 has species specificity. BX430 is used for chronic pain and cardiovascular disease.
For research use only. We do not sell to patients.
- CAS No.: 688309-70-8
- Formula: C15H15Br2N3O
- Molecular Weight:413.11
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Product Information
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
Chemical Information
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CAS No. 688309-70-8
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Molecular Weight 413.11
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Formula C15H15Br2N3O
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SMILES
O=C(NC1=CC=CN=C1)NC2=C(Br)C=C(C(C)C)C=C2Br
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Ase AR, et al. Identification and characterization of a selective allosteric antagonist of human P2X4 receptor channels. Mol Pharmacol. 2015 Apr;87(4):606-16. [Content Brief]
[2]. Sophocleous RA, et al. Pharmacological and genetic characterisation of the canine P2X4 receptor. Br J Pharmacol. 2020 Feb 4. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)