CB2R-IN-1
CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
For research use only. We do not sell to patients.
- CAS No.: 1257555-79-5
- Formula: C23H27F3N4O6S3
- Molecular Weight:608.67
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
CB2 0.9 nM (Ki) |
CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
-
CAS No. 1257555-79-5
-
Molecular Weight 608.67
-
Formula C23H27F3N4O6S3
-
SMILES
O=S(C(F)(F)F)(NCC1(CCC)CCN(S(=O)(C(N2S(=O)(C3=NC=CC=C3)=O)=CC4=C2C=CC=C4)=O)CC1)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)