ACG416B
Based on 1 Customer Validation
ACG416B (compound 18) is a potent inhibitor of ChoK (choline kinase) with an IC50 of 0.4 μM. ACG416B renders higher ChoK inhibitory and antiproliferative activities against the HT-29 human colon cancer cell.
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- Pureté: 98.99%
- CAS No.: 795316-15-3
- Formule: C38H36Br2N4
- Masse moléculaire:708.53
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Stockage:
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
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Activité biologique
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Chemical Information
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Solvant et solubilité
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
ChoK[1]
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HT-29 | IC50 |
2.2 μM
Compound: 18
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Antiproliferative activity was determined using HT-29 human colon cancer cell line
Antiproliferative activity was determined using HT-29 human colon cancer cell line
|
[PMID: 15481981] |
Chemical Information
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CAS No. 795316-15-3
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Appearance Solid
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Masse moléculaire 708.53
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Formule C38H36Br2N4
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Color White to off-white
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SMILES
CN(C1=CC=[N+](CC2=CC(C3=CC=CC(C[N+]4=CC=C(N(C)C5=CC=CC=C5)C=C4)=C3)=CC=C2)C=C1)C6=CC=CC=C6.[Br-].[Br-]
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Solvant et solubilité
DMSO : 100 mg/mL (141.14 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureté et documentation
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Fiche technique (265 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Instruction de manipulation (2659 KB)
Références
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 1.4114 mL | 7.0569 mL | 14.1137 mL | 35.2843 mL |
| 5 mM | 0.2823 mL | 1.4114 mL | 2.8227 mL | 7.0569 mL | |
| 10 mM | 0.1411 mL | 0.7057 mL | 1.4114 mL | 3.5284 mL | |
| 15 mM | 0.0941 mL | 0.4705 mL | 0.9409 mL | 2.3523 mL | |
| 20 mM | 0.0706 mL | 0.3528 mL | 0.7057 mL | 1.7642 mL | |
| 25 mM | 0.0565 mL | 0.2823 mL | 0.5645 mL | 1.4114 mL | |
| 30 mM | 0.0470 mL | 0.2352 mL | 0.4705 mL | 1.1761 mL | |
| 40 mM | 0.0353 mL | 0.1764 mL | 0.3528 mL | 0.8821 mL | |
| 50 mM | 0.0282 mL | 0.1411 mL | 0.2823 mL | 0.7057 mL | |
| 60 mM | 0.0235 mL | 0.1176 mL | 0.2352 mL | 0.5881 mL | |
| 80 mM | 0.0176 mL | 0.0882 mL | 0.1764 mL | 0.4411 mL | |
| 100 mM | 0.0141 mL | 0.0706 mL | 0.1411 mL | 0.3528 mL |
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