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Cat. No.: HY-N12399

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Aplithianines A

Aplithianines A is a potent inhibitor against J-PKA_cα with an IC₅₀ of 1 μM , and inhibits wild-type PKA with an IC₅₀ of 84 nM. Aplithianines A inhibits J-PKAcα catalytic activity by competitively binding to the ATP pocket.

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CAS No.: 3027425-38-0
Formule: C₁₃H₁₃N₇S
Masse moléculaire:299.35

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (269 KB)

Aplithianines A Chemical Structure

CAS No.: 3027425-38-0

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
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Activité biologique

Description

IC₅₀ & Target

1 μM (J-PKAcα)^[1]

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Chemical Information

CAS No. 3027425-38-0
Masse moléculaire 299.35
Formule C₁₃H₁₃N₇S
SMILES

CN1C=NC=C1C(SCC2)=CN2C3=NC=NC4=C3N=CN4
Structure Classification
- Alkaloids
- Other Alkaloids
Initial Source
- Microorganisms
Aplidium sp.
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (269 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Du L, et al. Discovery and Synthesis of a Naturally Derived Protein Kinase Inhibitor that Selectively Inhibits Distinct Classes of Serine/Threonine Kinases. J Nat Prod. 2023;86(10):2283-2293. IF: 5.1 Q1 B2 [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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Aplithianines A

Voir tous les produits spécifiques à Isoform PKA

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

Aplithianines A Related Classifications

HY-N12399 Related Classifications