CBR1-IN-3
Based on 1 Customer Validation
CBR1-IN-3 (compound 13h) is a potent inhibitor of carbonyl reductase 1 (CBR1), with IC50 value of 0.034 μM.
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- Pureté : 98.71%
- CAS No.: 891101-69-2
- Formule: C16H11ClN2O3
- Masse moléculaire:314.72
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Stockage:
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Activité biologique
Description
IC50 & Target
0.034 μM (CBR1)[1]
Cellular Effect
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CWR22R | IC50 |
3.3 μM
Compound: 2e
|
Antagonistic activity at AR in human 22Rv1 cells assessed as reduction in cell number by CCK8 assay
Antagonistic activity at AR in human 22Rv1 cells assessed as reduction in cell number by CCK8 assay
|
[PMID: 32847363] |
Chemical Information
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CAS No. 891101-69-2
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Appearance Solid
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Masse moléculaire 314.72
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Formule C16H11ClN2O3
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Color Light yellow to brown
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SMILES
O=C(C(C1=N)=CC2=C(O1)C(O)=CC=C2)NC3=CC=CC=C3Cl
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
4°C, sealed storage, away from moisture
* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
Pureté et documentation
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Fiche technique (270 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Instruction de manipulation (2659 KB)
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)