DS08701581
DS08701581 is an inhibitor of FER tyrosine kinase with IC50. DS08701581 has anti-tumor activity and oral activity.
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- CAS No.: 3074776-78-3
- Formule: C26H32N8O2
- Masse moléculaire:488.58
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| BaF3 | GI50 |
0.67 nM
Compound: 17c; DS08701581
|
Inhibition of cell viability in mouse BaF3 cells expressing FER incubated for 3 days by Cell Titer Glo assay
Inhibition of cell viability in mouse BaF3 cells expressing FER incubated for 3 days by Cell Titer Glo assay
|
[PMID: 39015278] |
| BaF3 | GI50 |
1000 nM
Compound: 17c; DS08701581
|
Inhibition of cell viability in mouse BaF3 cells incubated for 3 days by Cell Titer Glo assay
Inhibition of cell viability in mouse BaF3 cells incubated for 3 days by Cell Titer Glo assay
|
[PMID: 39015278] |
Chemical Information
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CAS No. 3074776-78-3
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Masse moléculaire 488.58
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Formule C26H32N8O2
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SMILES
O=C1NN=CC2=C(C#N)C(N[C@H]3[C@@H](N)CCCC3)=NC(NC4=CC=CC(N5C[C@H](C)O[C@H](C)C5)=C4)=C21
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)