GRL-03022
GRL-03022 is a potent, selective and non-covalent G protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 of 60 nM. GRL-03022 exhibits >16000-fold selectivity over GRK2 (IC50 > 1000 μM). GRL-03022 can be used for heart failure and cancer research.
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- Formule: C29H32N4O4
- Masse moléculaire:500.59
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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GRK2 >1000 μM (IC50) |
GRK5 60 nM (IC50) |
Chemical Information
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Masse moléculaire 500.59
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Formule C29H32N4O4
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SMILES
O=C(C1=CC2=C(NC(/C2=C\C3=C(C)C(C(N[C@@H](C)COC)=O)=C(C)N3)=O)C=C1)N[C@@H](C4=CC=CC=C4)C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
GRL-03022 Related Classifications
HY-179707 Related Classifications
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