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Cat. No.: HY-W934539

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Lenalidomide-amide-C8-Br

Lenalidomide-amide-C8-Br is an E3 ligase CRBN ligand-linker conjugate containing Lenalidomide (HY-A0003) and a linker. Lenalidomide-amide-C8-Br can be used to synthesize PROTAC PI3Kα/δ degrader-1 (HY-182083).

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CAS No.: 2580972-35-4
Formule: C₂₂H₂₈BrN₃O₄
Masse moléculaire:478.38

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Please store the product under the recommended conditions in the Certificate of Analysis.

Lenalidomide-amide-C8-Br Chemical Structure

CAS No.: 2580972-35-4

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Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Chemical Information
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Description

IC₅₀ & Target^[1]

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Chemical Information

CAS No. 2580972-35-4
Masse moléculaire 478.38
Formule C₂₂H₂₈BrN₃O₄
SMILES

O=C1NC(C(CC1)N2C(C3=C(C2)C(NC(CCCCCCCCBr)=O)=CC=C3)=O)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Hou Y, et al. Rational Design of Potent and Orally Efficacious PI3Kα/δ Degrader for PIK3CA Mutant Breast Cancer without Hyperglycemic Liability. J Med Chem. Published online March 8, 2026. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Lenalidomide-amide-C8-Br

Voir tous les produits spécifiques à Isoform E3 Ligase Ligand-Linker Conjugates