VU6077967
VU6077967 is a selective cannabinoid receptor 2 (CB2) agonist with an EC50 of 8.6 nM for rCB2. VU6077967 can be used for the research of neurological disease, suah as Alzheimer’s disease.
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- Formule: C26H36N2O6S
- Masse moléculaire:504.64
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
Description
IC50 & Target
[1]|
rat CB2-R 8.6 nM (EC50) |
In Vitro
VU6077967 (Compound 11d) potently activates rCB2 with an EC50 of 8.6 nM in a thallium flux assay[1].
VU6077967 inhibits arrestin and cAMP assay with an EC50 of 59 and 100 nM[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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Masse moléculaire 504.64
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Formule C26H36N2O6S
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SMILES
CC(CN(S(=O)(C1=CC=CC=C1)=O)C[C@H]([C@@H](NC(O[C@@H]2CCCOC2)=O)CC3=CC=CC=C3)O)C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)