BIM-23197
BIM-23197 is a selective SST2 (IC50 = 0.19 nM) agonist. BIM-23197 can effectively stimulate intracellular calcium mobilization in cells expressing SST2. BIM-23197 can be used for research on endocrine related conditions.
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- CAS. Nr.: 168016-90-8
- Formel: C57H81N13O13S3
- Molecular Weight:1252.53
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
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SSTR2 |
Chemical Information
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CAS. Nr. 168016-90-8
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Molecular Weight 1252.53
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Formel C57H81N13O13S3
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Sequence
{d-Phe(N-[[2-[4-(2-hydroxyethyl)-1-piperazinyl]ethyl]sulfonyl])}-Cys-Tyr-{d-Trp}-Lys-{Abu}-Cys-Thr-NH2 (Disulfide bridge: Cys2-Cys7)
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Sequence Shortening
{d-Phe(N-[[2-[4-(2-hydroxyethyl)-1-piperazinyl]ethyl]sulfonyl])}-CY-{d-Trp}-K-{Abu}-CT-NH2 (Disulfide bridge: Cys2-Cys7)
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
[1]. Tulipano G, et al. Characterization of new selective somatostatin receptor subtype-2 (sst2) antagonists, BIM-23627 and BIM-23454. Effects of BIM-23627 on GH release in anesthetized male rats after short-term high-dose dexamethasone treatment. Endocrinology. 2002 Apr;143(4):1218-24. [Content Brief]
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)