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Cat. No.: HY-123460

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BN-81674

BN-81674 is a somatostatin analogue and a selective antagonist of the non-peptide human somatostatin sst₃ receptor (K_i=0.92 nM). In addition, BN-81674 reversed the inhibition of cyclic AMP accumulation induced by 1 nM somatostatin through the sst₃ receptor with an IC₅₀ value of 0.84 nM. BN-81674 can be used in cancer research.

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CAS No.: 252278-73-2
Formule: C₃₀H₃₈N₄
Masse moléculaire:454.65

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (272 KB)

BN-81674 Chemical Structure

CAS No.: 252278-73-2

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

IC₅₀ & Target^[1]

SSTR3

0.92 nM (Ki)

Voir tous les produits spécifiques à Isoform Somatostatin Receptor :

Chemical Information

CAS No. 252278-73-2
Masse moléculaire 454.65
Formule C₃₀H₃₈N₄
SMILES

CCCCCC1(N[C@H](CC2=C1NC3=C2C=CC=C3)C4=NC=C(N4)C5=CC=CC=C5)CCCCC
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (272 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Poitout L, et al. Identification of potent non-peptide somatostatin antagonists with sst3 selectivity[J]. Journal of medicinal chemistry, 2001, 44(18): 2990-3000. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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BN-81674

Voir tous les produits spécifiques à Isoform Somatostatin Receptor

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

BN-81674 Related Classifications

HY-123460 Related Classifications