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Cat. No.: HY-121545

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CB-52

Name: CB-52
Brand: MedChemExpress
SKU: HY-121545
Price: 70.00 USD
Availability: InStock
Rating: 5 (1 reviews)

CB-52 is the ligand and neutral antagonist of CB2 cannabinoid receptor.

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CAS No.: 869376-90-9
Formule: C₂₆H₄₃NO₃
Masse moléculaire:417.62

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (263 KB)

CB-52 Chemical Structure

CAS No.: 869376-90-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- Cellular Effect
- In Vitro
- In Vivo
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

CB-52 is the ligand and neutral antagonist of CB2 cannabinoid receptor^[1].

Voir tous les produits spécifiques à Isoform Cannabinoid Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
RBL-2H3	IC₅₀	13 μM Compound: 52	Inhibition of anandamide membrane transporter in RBL-2H3 cells assessed as [14C]anandamide uptake Inhibition of anandamide membrane transporter in RBL-2H3 cells assessed as [14C]anandamide uptake	[PMID: 16279794]

In Vitro

CB-52 inhibits Forskolin (HY-15371)-induced cAMP formation by N18TG2 cells (IC₅₀: 450 nM) and hCB1-CHO cells (EC₅₀: 2600 nM)^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .

In Vivo

CB-52 (1 and 5 mg/kg, i.p.) decreases pain threshold to thermal stimulation in rats, and blocks WIN55,212-2 (2.5 mg/kg, i.p.) caused anti-nociceptive effect^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 869376-90-9
Masse moléculaire 417.62
Formule C₂₆H₄₃NO₃
SMILES

O=C(CCCCCCCCCCOC1=CC(O)=CC=C1CCCCCC)NC2CC2
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (263 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Cascio MG, et al. In vitro and in vivo pharmacology of synthetic olivetol- or resorcinol-derived cannabinoid receptor ligands. Br J Pharmacol. 2006 Oct;149(4):431-40. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

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MOQ

Minimum order quantity

100 mg

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