PD-135666
PD-135666 is a dipeptide inhibitor of cholecystokinin B (CCK B) receptors, binding to CCK B receptors in mouse cerebral cortex with IC50 of 0.1 nM. Its enantiomer, PD-140548, preferentially binds to CCK A receptors with IC50 of 2.8 nM in rat pancreas. PD-135666 exhibits anxiolytic effects in animal models.
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- CAS No.: 134557-41-8
- Formule: C33H39N3O5
- Masse moléculaire:557.68
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
IC50: 0.1 nM (CCK B Receptor)[1]
Chemical Information
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CAS No. 134557-41-8
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Masse moléculaire 557.68
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Formule C33H39N3O5
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SMILES
O=C(C[C@H](CC1=CC=CC=C1)NC([C@](NC(OC2C3CC4CC(CC2C4)C3)=O)(CC5=CNC6=C5C=CC=C6)C)=O)O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PD-135666 Related Classifications
HY-117839 Related Classifications
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