1. GPCR/G Protein
    Neuronal Signaling
  2. Dopamine Receptor
  3. CY 208-243

CY 208-243 

Cat. No.: HY-106094 Purity: 99.78%
Handling Instructions

CY 208-243 is a selective dopamine D1 receptor agonist which exhibits antiparkinsonian activity.

For research use only. We do not sell to patients.

CY 208-243 Chemical Structure

CY 208-243 Chemical Structure

CAS No. : 100999-26-6

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 287 In-stock
Estimated Time of Arrival: December 31
5 mg USD 285 In-stock
Estimated Time of Arrival: December 31
10 mg USD 485 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
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Based on 1 publication(s) in Google Scholar

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Description

CY 208-243 is a selective dopamine D1 receptor agonist which exhibits antiparkinsonian activity[1].

IC50 & Target

dopamine D1 receptor[1]

In Vivo

Pretreatment with CY 208-243 (2.5 mg/kg; s.c.) prevents the increase of DA release and metabolism induced by the D-1 antagonist, SCH 23390 (0.05 mg/kg; s.c.)[1].

Animal Model: Male Sprague-Dawley rats (180-200 g)[1]
Dosage: 2.5 mg/kg
Administration: Subcutaneous
Result: Prevented the increase of DA release and metabolism induced by the D-1 antagonist.
Molecular Weight

274.36

Formula

C₁₉H₁₈N₂

CAS No.

100999-26-6

SMILES

CN1[[email protected]@](C2)([H])[[email protected]@](C3=CC=CC=C3C1)([H])C4=CC=CC5=C4C2=CN5

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References
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Keywords:

CY 208-243Dopamine ReceptorDopamineD1Inhibitorinhibitorinhibit

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CY 208-243
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