1. GPCR/G Protein
    Neuronal Signaling
  2. mAChR
  3. Diphenmanil methylsulfate

Diphenmanil methylsulfate (Synonyms: Diphemanil mesylate)

Cat. No.: HY-16171 Purity: 99.83%
Handling Instructions

Diphemanil methylsulfate is a quaternary ammonium anticholinergic.

For research use only. We do not sell to patients.

Diphenmanil methylsulfate Chemical Structure

Diphenmanil methylsulfate Chemical Structure

CAS No. : 62-97-5

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Solution
10 mM * 1 mL in Water USD 66 In-stock
Estimated Time of Arrival: December 31
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ready for reconstitution
USD 66 In-stock
Estimated Time of Arrival: December 31
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10 mg USD 60 In-stock
Estimated Time of Arrival: December 31
50 mg USD 96 In-stock
Estimated Time of Arrival: December 31
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Description

Diphemanil methylsulfate is a quaternary ammonium anticholinergic. It binds muscarinic acetycholine receptors and thereby decreases secretory excretion of stomach acids as well as saliva and sweat. IC50 value: Target: mAChR Diphemanil Methylsulfate exerts its action by primarily binding the muscarinic M3 receptor. M3 receptors are located in the smooth muscles of the blood vessels, as well as in the lungs. This means they cause vasodilation and bronchoconstriction. They are also in the smooth muscles of the gastrointestinal tract (GIT), which help in increasing intestinal motility and dilating sphincters. The M3 receptors are also located in many glands which help to stimulate secretion in salivary glands and other glands of the body.

Molecular Weight

389.51

Formula

C21H27NO4S

CAS No.
Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

H2O : 16.67 mg/mL (42.80 mM; Need ultrasonic)

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Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5673 mL 12.8366 mL 25.6733 mL
5 mM 0.5135 mL 2.5673 mL 5.1347 mL
10 mM 0.2567 mL 1.2837 mL 2.5673 mL
*Please refer to the solubility information to select the appropriate solvent.
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Product Name:
Diphenmanil methylsulfate
Cat. No.:
HY-16171
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