DPP-4-IN-16
DPP-4-IN-16 (Compound 92) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor (IC50=0.8 nM). DPP-4-IN-16 inhibits DPP-4-mediated degradation of incretins (e.g., GLP-1 and GIP) to promote insulin secretion and reduce blood glucose. DPP-4-IN-16 is promising for research of type 2 diabetes.
For research use only. We do not sell to patients.
- Formula: C21H23BrN4O4
- Molecular Weight:475.34
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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DPP-4 0.8 nM (IC50) |
Chemical Information
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Molecular Weight 475.34
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Formula C21H23BrN4O4
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SMILES
[H]C1=C(N(C(N(C1=O)CC#CC)=O)N2CCC[C@@H](N)C2)CC3=C(Br)C=CC(C(O)=O)=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)