(E/Z)-Rivanicline
(E/Z)-Rivanicline ((E/Z)-RJR-2403, (E/Z)-Metanicotine) is the E/Z mixture of Rivanicline (HY-13225A). Rivanicline is a neuronal nicotinic receptor (neuronal nicotinic receptor) agonist that is highly selective for the α4β2 subtype, Ki is 26 nM, which is more than 1000 times more inhibitory than α7 receptor.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 538-79-4
- Fòrmula: C10H14N2
- Peso molecular:162.23
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Descripciòn
Cellular Effect
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| PC-12 | EC50 |
>1 mM
Compound: 15
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Compound was evaluated for functional potencies and efficacies at rat Nicotinic acetylcholine receptor subtype PC12 (ganglionic)
Compound was evaluated for functional potencies and efficacies at rat Nicotinic acetylcholine receptor subtype PC12 (ganglionic)
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[PMID: 9435889] |
Chemical Information
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No. CAS 538-79-4
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Peso molecular 162.23
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Fòrmula C10H14N2
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SMILES
CNCC/C=C/C1=CC=CN=C1
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Synonyms
(E/Z)-RJR-2403; (E/Z)-Metanicotine
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Structure Classification
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Initial Source
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
(E/Z)-Rivanicline Related Classifications
HY-13225E Related Classifications
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