Gartisertib (Standard)
Gartisertib (Standard) is the analytical standard of Gartisertib (HY-136270). This product is intended for research and analytical applications. Gartisertib (VX-803) is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. Gartisertib potently inhibits ATR-driven phosphorylated checkpoint Kinase-1 (Chk1) phosphorylation with an IC50 of 8 nM. Antitumor activity.
For research use only. We do not sell to patients.
- CAS No.: 1613191-99-3
- Formula: C25H29F2N9O3
- Molecular Weight:541.55
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Product Information
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Chemical Information
- Purity & Documentation
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Help & FAQs
Product Information
Information
Application
The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
Chemical Information
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CAS No. 1613191-99-3
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Molecular Weight 541.55
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Formula C25H29F2N9O3
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SMILES
O=C(C1=C2N=CC(F)=CN2N=C1N)NC3=C(N4CCC(C(N5CCN(C6COC6)CC5)=O)CC4)C(F)=CN=C3
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Synonyms
VX-803 (Standard); M4344 (Standard); ATR inhibitor 2 (Standard)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Gartisertib (Standard) Related Classifications
HY-136270R Related Classifications
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