EN10
EN10 is a ligand for the muscle-specific E3 ligase KLHL41, which can be used to synthesize PROTAC KBD-1 (HY-184151) targeting BRD4.
For research use only. We do not sell to patients.
- CAS No.: 2093466-80-7
- Formula: C21H23N3O
- Molecular Weight:333.43
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
KLHL41 |
In Vitro
Chemical Information
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CAS No. 2093466-80-7
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Molecular Weight 333.43
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Formula C21H23N3O
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SMILES
[C@@H]1(C2=CC=CC=C2)OCC[C@H]1CNCC3=CNN=C3C4=CC=CC=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
EN10 Related Classifications
HY-184150 Related Classifications
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Keywords
- EN10
- 2093466-80-7
- EN 10
- EN-10
- Ligands for E3 Ligase
- E1/E2/E3 Enzyme
- E3 ligase-recruiting Moiety
- E1 activating enzyme
- E2 conjugating enzyme
- E3 ligating enzyme
- Ubiquitin activating enzyme
- Ubiquitin conjugating enzyme
- Ubiquitin ligase
- androgen receptor
- rhabdomyosarcoma
- KLHL40
- RH30 human muscle rhabdomyosarcoma cells
- muscle cells
- KLHL41
- BRD4
- β-propeller domain
- GAPDH
- PROTAC
- Inhibitor
- inhibitor
- inhibit