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Referencia número: HY-121545

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CB-52

Name: CB-52
Brand: MedChemExpress
SKU: HY-121545
Price: 70.00 USD
Availability: InStock
Rating: 5 (1 reviews)

CB-52 is the ligand and neutral antagonist of CB2 cannabinoid receptor.

Para uso exclusivo en investigación. No vendemos a pacientes.

No. CAS: 869376-90-9
Fòrmula: C₂₆H₄₃NO₃
Peso molecular:417.62

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (263 KB)

CB-52 Chemical Structure

No. CAS: 869376-90-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica
- Descripciòn
- Cellular Effect
- In Vitro
- In Vivo
Chemical Information
Pureza y Documentación
Referencias
Calculators
Help & FAQs
Classifications
Bioz

Actividad biológica

Descripciòn

CB-52 is the ligand and neutral antagonist of CB2 cannabinoid receptor^[1].

Ver todos los productos específicos de isoformas Cannabinoid Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
RBL-2H3	IC₅₀	13 μM Compound: 52	Inhibition of anandamide membrane transporter in RBL-2H3 cells assessed as [14C]anandamide uptake Inhibition of anandamide membrane transporter in RBL-2H3 cells assessed as [14C]anandamide uptake	[PMID: 16279794]

In Vitro

CB-52 inhibits Forskolin (HY-15371)-induced cAMP formation by N18TG2 cells (IC₅₀: 450 nM) and hCB1-CHO cells (EC₅₀: 2600 nM)^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .

In Vivo

CB-52 (1 and 5 mg/kg, i.p.) decreases pain threshold to thermal stimulation in rats, and blocks WIN55,212-2 (2.5 mg/kg, i.p.) caused anti-nociceptive effect^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

No. CAS 869376-90-9
Peso molecular 417.62
Fòrmula C₂₆H₄₃NO₃
SMILES

O=C(CCCCCCCCCCOC1=CC(O)=CC=C1CCCCCC)NC2CC2
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (263 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Cascio MG, et al. In vitro and in vivo pharmacology of synthetic olivetol- or resorcinol-derived cannabinoid receptor ligands. Br J Pharmacol. 2006 Oct;149(4):431-40. [Content Brief]

Calculators

Calculadora de molaridad

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculadora de dilución

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

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MOQ

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100 mg

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