OMDM-3
OMDM-3 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki of 16.6 μM.
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- No. CAS: 616884-64-1
- Fòrmula: C29H43NO3
- Peso molecular:453.66
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
Ki: 16.6 μM (anandamide cellular uptake)[1]
OMDM-3 shows poor affinity for either CB1 (Ki=6.1 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-3 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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No. CAS 616884-64-1
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Peso molecular 453.66
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Fòrmula C29H43NO3
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SMILES
CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(N[C@@H](CC1=CC=C(O)C=C1)CO)=O
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Structure Classification
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Initial Source
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
OMDM-3 Related Classifications
HY-135880 Related Classifications
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