PTCA
Based on 1 Customer Validation
PTCA is a potent Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα) ligand with a pKi value of 7.2.
Para uso exclusivo en investigación. No vendemos a pacientes.
- Pureza: 99.72%
- No. CAS: 871326-47-5
- Fòrmula: C10H5Cl2NO2S
- Peso molecular:274.12
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Almacenamiento:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
Actividad biológica
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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No. CAS 871326-47-5
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Appearance Solid
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Peso molecular 274.12
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Fòrmula C10H5Cl2NO2S
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Color White to off-white
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SMILES
O=C(C1=CSC(C2=C(Cl)C=CC=C2Cl)=N1)O
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvente y solubilidad
DMSO : 100 mg/mL (364.80 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pureza y Documentación
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Ficha de datos (272 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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Instrucciones de manejo (2659 KB)
Referencias
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.6480 mL | 18.2402 mL | 36.4804 mL | 91.2009 mL |
| 5 mM | 0.7296 mL | 3.6480 mL | 7.2961 mL | 18.2402 mL | |
| 10 mM | 0.3648 mL | 1.8240 mL | 3.6480 mL | 9.1201 mL | |
| 15 mM | 0.2432 mL | 1.2160 mL | 2.4320 mL | 6.0801 mL | |
| 20 mM | 0.1824 mL | 0.9120 mL | 1.8240 mL | 4.5600 mL | |
| 25 mM | 0.1459 mL | 0.7296 mL | 1.4592 mL | 3.6480 mL | |
| 30 mM | 0.1216 mL | 0.6080 mL | 1.2160 mL | 3.0400 mL | |
| 40 mM | 0.0912 mL | 0.4560 mL | 0.9120 mL | 2.2800 mL | |
| 50 mM | 0.0730 mL | 0.3648 mL | 0.7296 mL | 1.8240 mL | |
| 60 mM | 0.0608 mL | 0.3040 mL | 0.6080 mL | 1.5200 mL | |
| 80 mM | 0.0456 mL | 0.2280 mL | 0.4560 mL | 1.1400 mL | |
| 100 mM | 0.0365 mL | 0.1824 mL | 0.3648 mL | 0.9120 mL |