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Referencia número: HY-120277

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TIPP

(Synonyms: H-Tyr-Tic-Phe-Phe-OH)

1 Cited Publications

Revisión del cliente

Based on 1 publication(s) in Google Scholar

TIPP is a potent and selective δ-opioid antagonist with a K_i value of 1.22 nM.

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No. CAS: 146369-65-5
Fòrmula: C₃₇H₃₈N₄O₆
Peso molecular:634.72

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (272 KB)

TIPP Chemical Structure

No. CAS: 146369-65-5

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Actividad biológica
- Descripciòn
- Cellular Effect
- Ensayo clínico
Chemical Information
Publications (1)
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Bioz

Actividad biológica

Descripciòn

TIPP is a potent and selective δ-opioid antagonist with a K_i value of 1.22 nM^[1].

Ver todos los productos específicos de isoformas Opioid Receptor :

Cellular Effect

Cell Line	Type	Value	Description	References
CHO	IC₅₀	22700 nM Compound: TIPP	Binding assay evaluated using DAMGO radioligand in CHO cells transfected with rat Opioid receptor mu 1 Binding assay evaluated using DAMGO radioligand in CHO cells transfected with rat Opioid receptor mu 1	[PMID: 11150176]
CHO	IC₅₀	5.8 nM Compound: TIPP	Binding assay evaluated using DPPE radioligand in CHO cells transfected with mouse Opioid receptor delta 1 Binding assay evaluated using DPPE radioligand in CHO cells transfected with mouse Opioid receptor delta 1	[PMID: 11150176]

Ensayo clínico

NCT Number	Sponsor	Condition	Start Date	Phase A549
NCT01329991	Plexxikon\|		2011-05	PHASE1

Chemical Information

No. CAS 146369-65-5
Peso molecular 634.72
Fòrmula C₃₇H₃₈N₄O₆
SMILES

O=C(N[C@@H](CC1=CC=CC=C1)C(N[C@H](C(O)=O)CC2=CC=CC=C2)=O)[C@H]3N(C([C@H](CC4=CC=C(O)C=C4)N)=O)CC5=CC=CC=C5C3
Synonyms

H-Tyr-Tic-Phe-Phe-OH
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Publications (1)

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Journal Impact Factor

Behav Pharmacol

2026 May 29.

Pureza y Documentación

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Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (272 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Schiller PW, et al. The TIPP opioid peptide family: development of delta antagonists, delta agonists, and mixed mu agonist/delta antagonists. Biopolymers. 1999;51(6):411-25. [Content Brief]

Calculators

Calculadora de molaridad

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Molecular Weight Molecular Weight

Calculadora de dilución

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Keywords

TIPP

1 Cited Publications

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Actividad biológica
- Descripciòn
- Ensayo clínico
Chemical Information
Publications (1)
Pureza y Documentación
Referencias

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TIPP

Publications Citing Use of MedChemExpress (MCE) TIPP

Ver todos los productos específicos de isoformas Opioid Receptor

Actividad biológica

Chemical Information

Publications (1)

Pureza y Documentación

Referencias

Calculators

Help & FAQs

TIPP Related Classifications

HY-120277 Related Classifications