1. Membrane Transporter/Ion Channel
  2. Potassium Channel
  3. Glisoxepide

Glisoxepide 

Cat. No.: HY-A0176
Handling Instructions

Glisoxepide, a sulphonamide derivative, is an orally available nonselective K(ATP) channel blocker, with antihyperglycemic activity and cardiovascular regulation effect.

For research use only. We do not sell to patients.

Glisoxepide Chemical Structure

Glisoxepide Chemical Structure

CAS No. : 25046-79-1

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Description

Glisoxepide, a sulphonamide derivative, is an orally available nonselective K(ATP) channel blocker, with antihyperglycemic activity and cardiovascular regulation effect[1][2][3].

IC50 & Target

K(ATP) channel[1]

In Vitro

Glisoxepide inhibits the uptake of bile acids into isolated rat hepatocytes[3].
Glisoxepide noncompetitively inhibits the cholate uptake with a Ki of 200 μM[3].

Molecular Weight

449.52

Formula

C₂₀H₂₇N₅O₅S

CAS No.

25046-79-1

SMILES

O=C(C1=NOC(C)=C1)NCCC2=CC=C(S(=O)(NC(NN3CCCCCC3)=O)=O)C=C2

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

GlisoxepidePotassium ChannelKcsAsulphonamidesulfonylureasK(ATP)potassiumchannelantihyperglycemicsulphonylureacardiovascularregulationInhibitorinhibitorinhibit

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