Pellotine
Pellotine is an alkaloid that can be isolated from Lophophora. Pellotine is the inverse agonist for 5-HT7 receptor with an EC50 of 291 nM. Pellotine exhibits good affinity to 5-HT1DR and 5-HT6R with Ki of 117 nM and 170 nM. Pellotine reduces intracellular cAMP levels, thereby reducing neuronal excitability and neurotransmitter release.
For research use only. We do not sell to patients.
- CAS No.: 19622-05-0
- Formula: C13H19NO3
- Molecular Weight:237.29
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
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5-HT7 Receptor |
Human 5-HT7 Receptor 291 nM (EC50) |
5-HT1D Receptor 117 nM (Ki) |
5-HT6 Receptor 170 nM (Ki) |
Chemical Information
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CAS No. 19622-05-0
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Molecular Weight 237.29
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Formula C13H19NO3
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SMILES
COC1=C(OC)C(O)=C(C(C)N(C)CC2)C2=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pellotine Related Classifications
HY-170908 Related Classifications
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