1. GPCR/G Protein
  2. Adenosine Receptor
  3. Inupadenant

Inupadenant (Synonyms: EOS-850)

Cat. No.: HY-137442
Handling Instructions

Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity.

For research use only. We do not sell to patients.

Inupadenant Chemical Structure

Inupadenant Chemical Structure

CAS No. : 2246607-08-7

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Description

Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].

IC50 & Target

A2A receptor[1]

Molecular Weight

604.65

Formula

C₂₅H₂₆F₂N₈O₄S₂

CAS No.
SMILES

O=C1SC(C2=NC(C3=CC=CO3)=NN2C(N)=N4)=C4N1CCN5CCN(C(C(F)=C6)=CC(OCC[[email protected]](C)=O)=C6F)CC5

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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  • Molarity Calculator

  • Dilution Calculator

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

InupadenantEOS-850EOS850EOS 850Adenosine ReceptorP1 receptororallyA2Abrain-penetrantInhibitorinhibitorinhibit

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Inupadenant
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HY-137442
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