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製品番号: HY-119060

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FP0429

FP0429 is a full mGlu4 agonist and partial mGlu8 agonist with EC₅₀ values of 48.3 μM and 56.2 μM, respectively.

商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。

CAS 番号: 870860-41-6
分子式: C₁₀H₁₂N₂O₇
分子量:272.21

保管条件:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (268 KB)

FP0429 構造式

CAS 番号: 870860-41-6

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価格（税別）

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性

製品説明

FP0429 is a full mGlu4 agonist and partial mGlu8 agonist with EC₅₀ values of 48.3 μM and 56.2 μM, respectively^[1].

mGluR アイソフォーム固有の製品をすべて表示 :

Cellular Effect

Cell Line	Type	Value	Description	References
HEK293	EC₅₀	>5000 μM Compound: 8a06, FP0429	Activity at rat mGluR2 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR2 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]
HEK293	EC₅₀	>5000 μM Compound: 8a06, FP0429	Activity at rat mGluR5 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR5 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]
HEK293	EC₅₀	378 μM Compound: 8a06, FP0429	Activity at rat mGluR6 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR6 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]
HEK293	EC₅₀	48.3 μM Compound: 8a06, FP0429	Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]
HEK293	EC₅₀	56.2 μM Compound: 8a06, FP0429	Activity at rat mGluR8 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR8 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]
HEK293	EC₅₀	>5000 μM Compound: 8a06, FP0429	Activity at rat mGluR1 receptor measured as intracellular calcium concentration in HEK293 cells Activity at rat mGluR1 receptor measured as intracellular calcium concentration in HEK293 cells	[PMID: 16828551]

化学情報

CAS 番号 870860-41-6
分子量 272.21
分子式 C₁₀H₁₂N₂O₇
SMILES

O=C(O)[C@H]1N(C[C@@](N)(C1)C(O)=O)C(/C=C/C(O)=O)=O
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.

純度とドキュメンテーション

バッチを選択:

純度: 99.98%

Assay: 99.98%

ee.: 99.98%

データシート (268 KB)
COA (2659 KB)
元素分析報告書 (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
取扱説明書 (2659 KB)

参考文献

[1]. Schann S, et al. Design and synthesis of APTCs (aminopyrrolidinetricarboxylic acids): identification of a new group III metabotropic glutamate receptor selective agonist. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4856-60. [Content Brief]

Calculators

モル濃度計算機

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

濃度濃度

体積体積

分子量分子量

希釈計算機

濃度 _(開始) × 体積 _(開始) = 濃度 _(終了) × 体積 _(終了)

濃度 _(開始) 濃度 _(開始)

体積 _(開始) 体積 _(開始)

濃度 _(終了) 濃度 _(終了)

体積 _(終了) 体積 _(終了)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

Minimum order quantity

100 mg

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生物活性
- 製品説明
化学情報
純度とドキュメンテーション
参考文献

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FP0429

mGluR アイソフォーム固有の製品をすべて表示

生物活性

化学情報

純度とドキュメンテーション

参考文献

Calculators

Help & FAQs

FP0429 関連分類

HY-119060 関連分類