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製品番号: HY-P1260

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FSLLRY-NH2

6 Cited Publications

カスタマーレビュー

Based on 6 publication(s) in Google Scholar

FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor.

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研究用途以外に使用した場合、当社は一切の責任を負いかねます。

純度: 99.89%
CAS 番号: 245329-02-6
分子式: C₃₉H₆₀N₁₀O₈
分子量:796.96

保管条件:

Sealed storage, away from moisture and light.

Powder -80°C, 2 years , -20°C, 1 year

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

FSLLRY-NH2 構造式

CAS 番号: 245329-02-6

容量

価格（税別）

在庫状況

数量

Amount: USD 0.00

* アイテムを追加する前、数量をご選択ください

Top Publications Citing

Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

生物活性

製品説明

FSLLRY-NH2 is a protease-activated receptor 2 (PAR2) inhibitor^[1].

IC₅₀ & Target

PAR2

Protease Activated Receptor (PAR) アイソフォーム固有の製品をすべて表示 :

体内実験

Treatment with FSLLRY-NH2 (50 μg per rat administered intranasally at 1 hour postresuscitation) significantly improves neurological outcome and reduces the number of degenerating hippocampal neurons after ACA (asphyxial CA)^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

化学情報

CAS 番号 245329-02-6
性状 Solid
分子量 796.96
分子式 C₃₉H₆₀N₁₀O₈
Color White to off-white
配列

Phe-Ser-Leu-Leu-Arg-Tyr-NH2
シーケンスの短縮

FSLLRY-NH2
輸送条件

Room temperature in continental US; may vary elsewhere.

保管条件

Sealed storage, away from moisture and light

Powder	-80°C	2 years
	-20°C	1 year

* In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Publications (6)

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Journal Impact Factor

J Immunother Cancer

Unveiling the mechanisms of CEBPD-orchestrated TAM polarization through RGS2/PAR2 pathway and its impact on ICB efficacy in clear cell renal cell carcinoma. [Abstract]

2025 Jul 13;13(7):e010898. PMID: 40659446
Brain Behav Immun

CD177 on neutrophils engages stress-related behavioral changes in male mice. [Abstract]

2024 Jun 12:120:403-412. PMID: 38871062
Biomolecules

PAR2 Participates in the Development of Cough Hypersensitivity in Guinea Pigs by Regulating TRPA1 Through PKC. [Abstract]

2025 Feb 1;15(2):208. PMID: 40001511
Cell Signal

Angiotensin II depends on hippo/YAP signaling to reprogram angiogenesis and promote liver fibrosis. [Abstract]

2024 Nov:123:111355. PMID: 39173854
BMC Musculoskelet Disord

Knockdown of PAR2 alleviates cancer-induced bone pain by inhibiting the activation of astrocytes and the ERK pathway. [Abstract]

2022 May 30;23(1):514. PMID: 35637468
Res Sq

2024 Sep 04.

溶剤 & 溶解度

体外:

DMSO : 100 mg/mL (125.48 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

View the Complete Stock Solution Preparation Table

Preparing Stock Solutions

View the Complete Stock Solution Preparation Table

Concentration Solvent Mass

1 mg

5 mg

10 mg

Concentration

Solvent

Mass

1 mM

1.2548 mL

6.2738 mL

12.5477 mL

5 mM

0.2510 mL

1.2548 mL

2.5095 mL

10 mM

0.1255 mL

0.6274 mL

1.2548 mL

Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.

Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

モル濃度計算機

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

濃度濃度

体積体積

分子量分子量

希釈計算機

濃度 _(開始) × 体積 _(開始) = 濃度 _(終了) × 体積 _(終了)

濃度 _(開始) 濃度 _(開始)

体積 _(開始) 体積 _(開始)

濃度 _(終了) 濃度 _(終了)

体積 _(終了) 体積 _(終了)

純度とドキュメンテーション

バッチを選択:

純度: 99.98%

Assay: 99.98%

ee.: 99.98%

データシート (272 KB)
SDS (394 KB)
- English - EN (394 KB)
- Français - FR (394 KB)
- Deutsch - DE (394 KB)
- Norwegian - NO (394 KB)
- Español - ES (394 KB)
- Swedish - SV (394 KB)
- Italian - IT (394 KB)
- Korean - KR (394 KB)
- Portuguese - PT (394 KB)
COA (2659 KB)
元素分析報告書 (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
取扱説明書 (2659 KB)

参考文献

[1]. Umut Ocak, et al. FSLLRY-NH2 Improves Neurological Outcome After Cardiac Arrest in Rats. Turk Neurosurg. 2020;30(2):244-251. [Content Brief]

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg
DMSO	1 mM	1.2548 mL	6.2738 mL	12.5477 mL	31.3692 mL
	5 mM	0.2510 mL	1.2548 mL	2.5095 mL	6.2738 mL
	10 mM	0.1255 mL	0.6274 mL	1.2548 mL	3.1369 mL
	15 mM	0.0837 mL	0.4183 mL	0.8365 mL	2.0913 mL
	20 mM	0.0627 mL	0.3137 mL	0.6274 mL	1.5685 mL
	25 mM	0.0502 mL	0.2510 mL	0.5019 mL	1.2548 mL
	30 mM	0.0418 mL	0.2091 mL	0.4183 mL	1.0456 mL
	40 mM	0.0314 mL	0.1568 mL	0.3137 mL	0.7842 mL
	50 mM	0.0251 mL	0.1255 mL	0.2510 mL	0.6274 mL
	60 mM	0.0209 mL	0.1046 mL	0.2091 mL	0.5228 mL
	80 mM	0.0157 mL	0.0784 mL	0.1568 mL	0.3921 mL
	100 mM	0.0125 mL	0.0627 mL	0.1255 mL	0.3137 mL

Keywords

FSLLRY-NH2

6 Cited Publications

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100 mg

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FSLLRY-NH2

Peptide Library

Coagulation and Anti-coagulation Compound Library

Membrane Protein-targeted Compound Library

Membrane Receptor-targeted Compound Library

Bioactive Compound Library Max

MCE Bioactive Compound Library

Bioactive Compound Library

High-Throughput Bioactive Compound Library

Lactylation Compound Library

GPCR/G Protein Compound Library

Peptide Compound Library

MedChemExpress（MCE）の使用を引用している文献 FSLLRY-NH2

Protease Activated Receptor (PAR) アイソフォーム固有の製品をすべて表示

生物活性

化学情報

Publications (6)

溶剤 & 溶解度

純度とドキュメンテーション

参考文献

Help & FAQs

Complete Stock Solution Preparation Table

FSLLRY-NH2

Peptide Library

Coagulation and Anti-coagulation Compound Library

Membrane Protein-targeted Compound Library

Membrane Receptor-targeted Compound Library

Bioactive Compound Library Max

MCE Bioactive Compound Library

Bioactive Compound Library

High-Throughput Bioactive Compound Library

Lactylation Compound Library

GPCR/G Protein Compound Library

Peptide Compound Library

MedChemExpress（MCE）の使用を引用している文献 FSLLRY-NH2

Protease Activated Receptor (PAR) アイソフォーム固有の製品をすべて表示

生物活性

化学情報

Publications (6)

溶剤 & 溶解度

純度とドキュメンテーション

参考文献

Help & FAQs

Complete Stock Solution Preparation Table

FSLLRY-NH2 関連分類

HY-P1260 関連分類