PTCA
Based on 1 Customer Validation
PTCA is a potent Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα) ligand with a pKi value of 7.2.
商品は「研究用試薬」です。人や動物の医療用・臨床診断用・食品用の製品ではありません。
研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 純度: 99.72%
- CAS 番号: 871326-47-5
- 分子式: C10H5Cl2NO2S
- 分子量:274.12
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保管条件:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
生物活性
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
化学情報
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CAS 番号 871326-47-5
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性状 Solid
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分子量 274.12
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分子式 C10H5Cl2NO2S
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Color White to off-white
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SMILES
O=C(C1=CSC(C2=C(Cl)C=CC=C2Cl)=N1)O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
溶剤 & 溶解度
DMSO : 100 mg/mL (364.80 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
純度とドキュメンテーション
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データシート (272 KB)
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SDS (393 KB)
- English - EN (393 KB)
- Français - FR (393 KB)
- Deutsch - DE (393 KB)
- Norwegian - NO (393 KB)
- Español - ES (393 KB)
- Swedish - SV (393 KB)
- Italian - IT (393 KB)
- Korean - KR (393 KB)
- Portuguese - PT (393 KB)
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取扱説明書 (2659 KB)
参考文献
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.6480 mL | 18.2402 mL | 36.4804 mL | 91.2009 mL |
| 5 mM | 0.7296 mL | 3.6480 mL | 7.2961 mL | 18.2402 mL | |
| 10 mM | 0.3648 mL | 1.8240 mL | 3.6480 mL | 9.1201 mL | |
| 15 mM | 0.2432 mL | 1.2160 mL | 2.4320 mL | 6.0801 mL | |
| 20 mM | 0.1824 mL | 0.9120 mL | 1.8240 mL | 4.5600 mL | |
| 25 mM | 0.1459 mL | 0.7296 mL | 1.4592 mL | 3.6480 mL | |
| 30 mM | 0.1216 mL | 0.6080 mL | 1.2160 mL | 3.0400 mL | |
| 40 mM | 0.0912 mL | 0.4560 mL | 0.9120 mL | 2.2800 mL | |
| 50 mM | 0.0730 mL | 0.3648 mL | 0.7296 mL | 1.8240 mL | |
| 60 mM | 0.0608 mL | 0.3040 mL | 0.6080 mL | 1.5200 mL | |
| 80 mM | 0.0456 mL | 0.2280 mL | 0.4560 mL | 1.1400 mL | |
| 100 mM | 0.0365 mL | 0.1824 mL | 0.3648 mL | 0.9120 mL |