UVI3502
UVI3502 is a cannabinoid receptor 1 (CB1) antagonist with an IC50 value of 4641 nM for CB1 and approximately 16200 nM for CB2. UVI3502 blocks Gi/o protein coupling induced by the agonist CP55,940. UVI3502 is promising for research of endocannabinoid system-related diseases in the central nervous system (such as cognitive impairment and neurodegenerative diseases).
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- 分子式: C25H24N2O6
- 分子量:448.47
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
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CB1 4641 nM (IC50) |
CB2 16200 nM (IC50) |
化学情報
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分子量 448.47
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分子式 C25H24N2O6
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SMILES
COC1=CC2=C(N(C(OCC)=O)C(C(C=C(C)C=C3)=C3NC/4=O)=C2C4=C\C(OCC)=O)C=C1
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)