KAT2A/B ligand 1
Based on 1 Customer Validation
KAT2A/B ligand 1 (compound 32a) is a KAT2A/B ligand. KAT2A/B ligand 1 can be used as a target protein ligand for the synthesis of AUR1545 (HY-173158).
For research use only. We do not sell to patients.
- Purity: 99.07%
- CAS No.: 2254066-18-5
- Formula: C18H21BrN4O3
- Molecular Weight:421.29
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Storage:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
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Biological Activity
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Chemical Information
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Solvent & Solubility
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Description
IC50 & Target
[1]|
GCN5/PCAF |
Chemical Information
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CAS No. 2254066-18-5
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Appearance Solid
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Molecular Weight 421.29
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Formula C18H21BrN4O3
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Color Light yellow to yellow
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SMILES
O=C(O)C1=CC=C([C@@H]2CN(C)C[C@H](NC(C=NN3C)=C(Br)C3=O)C2)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
Solvent & Solubility
In Vitro:
DMSO : 100 mg/mL (237.37 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Purity & Documentation
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Data Sheet (270 KB)
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SDS (252 KB)
- English - EN (252 KB)
- Français - FR (252 KB)
- Deutsch - DE (252 KB)
- Norwegian - NO (252 KB)
- Español - ES (252 KB)
- Swedish - SV (252 KB)
- Italian - IT (252 KB)
- Korean - KR (252 KB)
- Portuguese - PT (252 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.3737 mL | 11.8683 mL | 23.7366 mL | 59.3415 mL |
| 5 mM | 0.4747 mL | 2.3737 mL | 4.7473 mL | 11.8683 mL | |
| 10 mM | 0.2374 mL | 1.1868 mL | 2.3737 mL | 5.9342 mL | |
| 15 mM | 0.1582 mL | 0.7912 mL | 1.5824 mL | 3.9561 mL | |
| 20 mM | 0.1187 mL | 0.5934 mL | 1.1868 mL | 2.9671 mL | |
| 25 mM | 0.0949 mL | 0.4747 mL | 0.9495 mL | 2.3737 mL | |
| 30 mM | 0.0791 mL | 0.3956 mL | 0.7912 mL | 1.9781 mL | |
| 40 mM | 0.0593 mL | 0.2967 mL | 0.5934 mL | 1.4835 mL | |
| 50 mM | 0.0475 mL | 0.2374 mL | 0.4747 mL | 1.1868 mL | |
| 60 mM | 0.0396 mL | 0.1978 mL | 0.3956 mL | 0.9890 mL | |
| 80 mM | 0.0297 mL | 0.1484 mL | 0.2967 mL | 0.7418 mL | |
| 100 mM | 0.0237 mL | 0.1187 mL | 0.2374 mL | 0.5934 mL |
KAT2A/B ligand 1 Related Classifications
HY-W1122565 Related Classifications
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