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Cat. No.: HY-W1122565

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KAT2A/B ligand 1

KAT2A/B ligand 1 (compound 32a) is a KAT2A/B ligand. KAT2A/B ligand 1 can be used as a target protein ligand for the synthesis of AUR1545 (HY-173158).

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CAS No.: 2254066-18-5
Formule: C₁₈H₂₁BrN₄O₃
Masse moléculaire:421.29

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Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (266 KB)

KAT2A/B ligand 1 Chemical Structure

CAS No.: 2254066-18-5

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
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Description

KAT2A/B ligand 1 (compound 32a) is a KAT2A/B ligand. KAT2A/B ligand 1 can be used as a target protein ligand for the synthesis of AUR1545 (HY-173158)^[1].

IC₅₀ & Target^[1]

GCN5/PCAF

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Chemical Information

CAS No. 2254066-18-5
Masse moléculaire 421.29
Formule C₁₈H₂₁BrN₄O₃
SMILES

O=C(O)C1=CC=C([C@@H]2CN(C)C[C@H](NC(C=NN3C)=C(Br)C3=O)C2)C=C1
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Select Batch:

Pureté: 99.98%

Assay: 99.98%

ee.: 99.98%

Fiche technique (266 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instruction de manipulation (2659 KB)

Références

[1]. Neef J, et al. Discovery and Optimization of Orally Bioavailable Heterobifunctional Degraders of KAT2A/B for the Treatment of Cancer. J Med Chem. 2026 Feb 26;69(4):4548-4566. [Content Brief]

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Calculateur de dilution

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Concentration _(final) Concentration _(final)

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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- IC₅₀ & Target
Chemical Information
Pureté et documentation
Références

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KAT2A/B ligand 1

Voir tous les produits spécifiques à Isoform Histone Acetyltransferase

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

KAT2A/B ligand 1 Related Classifications

HY-W1122565 Related Classifications