TP003
Based on 1 Customer Validation
TP003 is a non-selective benzodiazepine site agonist with EC50s of 20.3, 10.6, 3.24, 5.64 nM for α1β2γ2, α2β3γ2, α3β3γ2, α5β2γ2, respectively. TP003 induces anxiolysis via α2GABAA receptors.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- Purity : 98.09%
- CAS No.: 628690-75-5
- 화학식: C23H16F3N3O
- 분자량:407.39
-
보관:Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
-
용액&용해도
- 순도&문서
- References
-
Help & FAQs
-
HY-B0009
FlumazenilGABA Receptor Antagonist -
HY-W001692
OcinaplonGABAA receptor Modulator -
HY-103476
Ro15-4513Benzodiazepine Receptor Antagonist -
HY-B0009R
Flumazenil (Standard)GABA Receptor Antagonist -
HY-116622
α5IAGABAA Receptor Agonist -
HY-B0007
BaclofenGABABR Agonist -
HY-19567
PK 11195Parasite Inhibitor -
HY-107994
Aminooxyacetic acid hemihydrochlorideGABA Receptor Inhibitor -
HY-100813
SaclofenGABAB Receptor Antagonist -
HY-103504
(S)-SNAP5114GABA Transporter Inhibitor -
HY-103531
CGP52432GABAB Antagonist -
HY-100798
PhaclofenGABAB Receptor Antagonist
Biological Activity
제품 설명
Chemical Information
-
CAS No. 628690-75-5
-
Appearance Solid
-
분자량 407.39
-
화학식 C23H16F3N3O
-
Color White to off-white
-
SMILES
N#CC1=CC(F)=CC=C1C2=CC(C3=CN=C4C(F)=C(C(C)(O)C)C=CN43)=CC=C2F
-
선적
Room temperature in continental US; may vary elsewhere.
-
보관
Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
용액&용해도
In Vitro:
DMSO : 100 mg/mL (245.47 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
순도&문서
-
Data Sheet (271 KB)
-
SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
-
Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 2.4547 mL | 12.2733 mL | 24.5465 mL | 61.3663 mL |
| 5 mM | 0.4909 mL | 2.4547 mL | 4.9093 mL | 12.2733 mL | |
| 10 mM | 0.2455 mL | 1.2273 mL | 2.4547 mL | 6.1366 mL | |
| 15 mM | 0.1636 mL | 0.8182 mL | 1.6364 mL | 4.0911 mL | |
| 20 mM | 0.1227 mL | 0.6137 mL | 1.2273 mL | 3.0683 mL | |
| 25 mM | 0.0982 mL | 0.4909 mL | 0.9819 mL | 2.4547 mL | |
| 30 mM | 0.0818 mL | 0.4091 mL | 0.8182 mL | 2.0455 mL | |
| 40 mM | 0.0614 mL | 0.3068 mL | 0.6137 mL | 1.5342 mL | |
| 50 mM | 0.0491 mL | 0.2455 mL | 0.4909 mL | 1.2273 mL | |
| 60 mM | 0.0409 mL | 0.2046 mL | 0.4091 mL | 1.0228 mL | |
| 80 mM | 0.0307 mL | 0.1534 mL | 0.3068 mL | 0.7671 mL | |
| 100 mM | 0.0245 mL | 0.1227 mL | 0.2455 mL | 0.6137 mL |
TP003 Related Classifications
HY-103512 Related Classifications
Powered by Bioz