1. Metabolic Enzyme/Protease
    Autophagy
    Apoptosis
  2. Dipeptidyl Peptidase
    Autophagy
    Ferroptosis
  3. Linagliptin-d4

Linagliptin-d4  (Synonyms: BI 1356-d4)

Cat. No.: HY-10284S
Handling Instructions

Linagliptin-d4 is deuterium labeled Linagliptin. Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.

For research use only. We do not sell to patients.

Linagliptin-d4 Chemical Structure

Linagliptin-d4 Chemical Structure

CAS No. : 2140263-92-7

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1 mg USD 450 In-stock
Estimated Time of Arrival: December 31
5 mg USD 1450 In-stock
Estimated Time of Arrival: December 31
10 mg USD 2400 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

Linagliptin-d4 is deuterium labeled Linagliptin. Linagliptin is a highly potent, selective DPP-4 inhibitor with IC50 of 1 nM.

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

476.57

Formula

C25H24D4N8O2

CAS No.
SMILES

CC#CCN1C2=C(N(C(N(C2=O)CC3=NC4=C(C=CC=C4)C(C)=N3)=O)C)N=C1N5C([2H])([2H])[[email protected]@H](CCC5([2H])[2H])N

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
References
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Linagliptin-d4
Cat. No.:
HY-10284S
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