MDA77
MDA77 is a CB2 inverse agonist with an EC50 of 5.82 nM, showing selectivity for human CB2 and no activity on CB1.
For research use only. We do not sell to patients.
- CAS No.: 1103774-21-5
- Formula: C21H23N3O3
- Molecular Weight:365.43
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
263 nM
Compound: 16, MDA77
|
Inverse agonist activity at human recombinant CB1 receptor expressed CHO cells membrane by [35S]GTPgamma binding assay
Inverse agonist activity at human recombinant CB1 receptor expressed CHO cells membrane by [35S]GTPgamma binding assay
|
[PMID: 19115816] |
| CHO | EC50 |
5.8 nM
Compound: 16, MDA77
|
Inverse agonist activity at human recombinant CB2 receptor expressed CHO cells membrane by [35S]GTPgamma binding assay
Inverse agonist activity at human recombinant CB2 receptor expressed CHO cells membrane by [35S]GTPgamma binding assay
|
[PMID: 19115816] |
Chemical Information
-
CAS No. 1103774-21-5
-
Molecular Weight 365.43
-
Formula C21H23N3O3
-
SMILES
O=C(N/N=C1C(N(CCCCC)C2=C\1C=CC(OC)=C2)=O)C3=CC=CC=C3
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MDA77 Related Classifications
HY-113885 Related Classifications
Powered by Bioz